CFAMM00131060 |
CHEMBL213291 |
Bioactive |
SureCN12306982 |
CFAMM00131151 |
CHEMBL2021559 |
Bioactive |
(4R,7S,10S,13R,16S,19R)-19-amino-N-[(2S)-1-amino-3-naphthalen-2-yl-1-oxopropan-2-yl]-7,16-dibenzyl-13-[methyl(naphthalene-2-carbonyl)amino]-6,9,12,15,18-pentaoxo-10-[[4-[(propan-2-ylamino)methyl]phenyl]methyl]-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide |
CFAMM00130999 |
CHEMBL538451 |
Bioactive |
(4R,7S,10S,13R,16S,19S)-10-(4-aminobutyl)-19-[[(2S)-2-amino-3-(4-carbamoylphenyl)propanoyl]amino]-N-[(2S)-1-amino-3-naphthalen-2-yl-1-oxopropan-2-yl]-7,16-dibenzyl-13-[methyl(naphthalene-2-carbonyl)amino]-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide |
CFAMM00131027 |
CHEMBL212434 |
Bioactive |
SureCN12306946 |
CFAMM00130992 |
CHEMBL104348 |
Bioactive |
3-[[[3,5-bis(trifluoromethyl)benzoyl]-methylamino]-(naphthalen-2-ylmethyl)amino]-N-[(3R)-2-oxoazepan-3-yl]propanamide |
CFAMM00131005 |
CHEMBL428055 |
Bioactive |
SureCN12306968 |
CFAMM00130985 |
CHEMBL399465 |
Bioactive |
SureCN12306970 |
CFAMM00130998 |
CHEMBL583285 |
Bioactive |
(2S)-2-[[(3S)-2-[(2S)-2-amino-3-[4-[2-(4-phenylphenyl)ethylcarbamoyl]phenyl]propanoyl]-3,4-dihydro-1H-isoquinoline-3-carbonyl]amino]-3-phenylpropanoic acid |
CFAMM00131100 |
CHEMBL493465 |
Bioactive |
3-cyano-N-[[4-fluoro-3-[3-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]phenyl]methyl]benzamide |
CFAMM00131026 |
CHEMBL446757 |
Bioactive |
(3S)-N-[(2R)-3-(4-fluorophenyl)-1-[(2S)-4-[(2S)-1-(methylamino)-3-naphthalen-2-yl-1-oxopropan-2-yl]-3-oxo-2-propylpiperazin-1-yl]-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide |
CFAMM00130978 |
CHEMBL448410 |
Bioactive |
(2R)-N-[(2R)-3-(4-fluorophenyl)-1-[(2S)-4-[(2S)-1-(methylamino)-3-naphthalen-2-yl-1-oxopropan-2-yl]-3-oxo-2-propylpiperazin-1-yl]-1-oxopropan-2-yl]piperidine-2-carboxamide |
CFAMM00131157 |
CHEMBL63400 |
Bioactive |
N,N-diethyl-4-[[8-[2-(4-fluorophenyl)ethyl]-8-azabicyclo[3.2.1]octan-3-ylidene]-phenylmethyl]benzamide |
CFAMM00130942 |
CHEMBL280587 |
Bioactive |
N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-2-[(E)-2-naphthalen-2-ylethenyl]benzamide |
CFAMM00130991 |
CHEMBL251161 |
Bioactive |
SureCN12306967 |
CFAMM00130997 |
CHEMBL239923 |
Bioactive |
AGN-PC-04T15F |
CFAMM00131072 |
CHEMBL452710 |
Bioactive |
(2S)-2-[(3S)-4-[(2R)-3-(4-fluorophenyl)-2-[[2-(methylamino)acetyl]amino]propanoyl]-2-oxo-3-propylpiperazin-1-yl]-N-methyl-3-naphthalen-2-ylpropanamide |
CFAMM00130951 |
CHEMBL430397 |
Bioactive |
SureCN12306966 |
CFAMM00130990 |
CHEMBL251160 |
Bioactive |
CHEMBL251160 |
CFAMM00131064 |
CHEMBL2206329 |
Bioactive |
(2S)-2-[[(2S)-2-[[2-[(2S)-2-amino-3-[4-(2-naphthalen-1-ylethylcarbamoyl)phenyl]propanoyl]-3,4-dihydro-1H-isoquinoline-3-carbonyl]amino]-3-phenylpropanoyl]amino]-3-phenylpropanoic acid |
CFAMM00131092 |
CHEMBL499884 |
Bioactive |
CHEMBL499884 |
CFAMM00131105 |
CHEMBL200788 |
Bioactive |
AGN-PC-00A9WU |
CFAMM00131122 |
CHEMBL567288 |
Bioactive |
AGN-PC-00CQH0 |
CFAMM00130983 |
CHEMBL103979 |
Bioactive |
N-methyl-N-[(E,2R)-1-naphthalen-2-yl-5-oxo-5-[[(3R)-2-oxoazepan-3-yl]amino]pent-3-en-2-yl]-3,5-bis(trifluoromethyl)benzamide |
CFAMM00131135 |
CHEMBL466380 |
Bioactive |
(2S)-2-[(3S)-4-[(2R)-2-acetamido-3-(4-fluorophenyl)propanoyl]-2-oxo-3-propylpiperazin-1-yl]-N-methyl-3-naphthalen-2-ylpropanamide |
CFAMM00131148 |
CHEMBL506762 |
Bioactive |
N-[(2R)-3-(4-fluorophenyl)-1-[(2S)-4-[(2S)-1-(methylamino)-3-naphthalen-2-yl-1-oxopropan-2-yl]-3-oxo-2-propylpiperazin-1-yl]-1-oxopropan-2-yl]piperidine-4-carboxamide |
CFAMM00131128 |
CHEMBL296397 |
Bioactive |
2-[3,5-bis(trifluoromethyl)phenyl]-N-[4-[4-(4-fluorophenyl)piperidin-1-yl]-1-phenylcyclohexyl]propanamide |
CFAMM00131155 |
CHEMBL426863 |
Bioactive |
AGN-PC-00ESCP |
CFAMM00131030 |
CHEMBL209550 |
Bioactive |
SureCN12306981 |
CFAMM00131070 |
CHEMBL583486 |
Bioactive |
(2S)-2-[[(2S)-2-[[(3S)-2-[(2S)-2-amino-3-[4-[2-(4-phenylphenyl)ethylcarbamoyl]phenyl]propanoyl]-3,4-dihydro-1H-isoquinolin-3-yl]methylamino]-3-cyclohexylpropanoyl]amino]-3-phenylpropanoic acid |
CFAMM00131001 |
CHEMBL281764 |
Bioactive |
Tabimorelin |
CFAMM00131153 |
CHEMBL572542 |
Bioactive |
(2S)-2-[[(2S)-2-[[(3S)-2-[(2S)-2-amino-3-[4-[2-(4-phenylphenyl)ethylcarbamoyl]phenyl]propanoyl]-3,4-dihydro-1H-isoquinoline-3-carbonyl]amino]-3-phenylpropanoyl]amino]-3-phenylpropanoic acid |
CFAMM00131042 |
CHEMBL51926 |
Bioactive |
2-[3,5-bis(trifluoromethyl)phenyl]-N-[4-(4-methylpiperidin-1-yl)-1-phenylcyclohexyl]propanamide |
CFAMM00131096 |
CHEMBL583485 |
Bioactive |
(2S)-2-[[(2S)-2-[[(3S)-2-[(2S)-2-amino-3-[4-[2-(4-phenylphenyl)ethylcarbamoyl]phenyl]propanoyl]-3,4-dihydro-1H-isoquinolin-3-yl]methylamino]-3-phenylpropanoyl]amino]-3-phenylpropanoic acid |
CFAMM00130974 |
CHEMBL453734 |
Bioactive |
2-amino-N-[(2R)-3-(4-fluorophenyl)-1-[(2S)-4-[(2S)-1-(methylamino)-3-naphthalen-2-yl-1-oxopropan-2-yl]-3-oxo-2-propylpiperazin-1-yl]-1-oxopropan-2-yl]-2-methylpropanamide |
CFAMM00131014 |
CHEMBL215594 |
Bioactive |
SureCN12306950 |
CFAMM00131102 |
CHEMBL250388 |
Bioactive |
CHEMBL250388 |
CFAMM00130967 |
CHEMBL507876 |
Bioactive |
N-[(2R)-3-(4-fluorophenyl)-1-[(2S)-4-[(2S)-1-(methylamino)-3-naphthalen-2-yl-1-oxopropan-2-yl]-3-oxo-2-propylpiperazin-1-yl]-1-oxopropan-2-yl]-2,2-dimethylpropanamide |
CFAMM00131132 |
CHEMBL2206330 |
Bioactive |
(2S)-2-[[(2S)-2-[[2-[(2S)-2-amino-3-[4-(2-naphthalen-2-ylethylcarbamoyl)phenyl]propanoyl]-3,4-dihydro-1H-isoquinoline-3-carbonyl]amino]-3-phenylpropanoyl]amino]-3-phenylpropanoic acid |
CFAMM00130946 |
CHEMBL504349 |
Bioactive |
(2S)-2-[(3S)-4-[(2R)-3-(4-fluorophenyl)-2-[[(2S)-2-(methylamino)propanoyl]amino]propanoyl]-2-oxo-3-propylpiperazin-1-yl]-N-methyl-3-naphthalen-2-ylpropanamide |
CFAMM00131074 |
CHEMBL257702 |
Bioactive |
N-[2-[[(3R)-1-[(4-fluorophenyl)methyl]pyrrolidin-3-yl]amino]-2-oxoethyl]-3-(trifluoromethyl)benzamide |
CFAMM00131125 |
CHEMBL212928 |
Bioactive |
(2S)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-2-(4-fluorophenyl)-4-spiro[1,2-dihydroindene-3,4'-piperidine]-1'-ylbutanamide |
CFAMM00130973 |
CHEMBL2021544 |
Bioactive |
(4R,7S,10S,13S,16S,19R)-19-amino-N-[(2S)-1-amino-3-naphthalen-2-yl-1-oxopropan-2-yl]-7,16-dibenzyl-13-[methyl(naphthalene-2-carbonyl)amino]-6,9,12,15,18-pentaoxo-10-[[4-[(propan-2-ylamino)methyl]phenyl]methyl]-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide |
CFAMM00131088 |
CHEMBL2022530 |
Bioactive |
N-[2-[(2S)-2-cyano-4,4-difluoropyrrolidin-1-yl]-2-oxoethyl]naphthalene-1-carboxamide |
CFAMM00131165 |
CHEMBL248421 |
Bioactive |
SureCN5117385 |
CFAMM00130937 |
CHEMBL2031990 |
Bioactive |
N-[[(3R)-1-[6,6-bis(4-fluorophenyl)hexanoyl]pyrrolidin-3-yl]methyl]-3,5-bis(trifluoromethyl)benzamide |
CFAMM00131131 |
CHEMBL423917 |
Bioactive |
2-phenyl-N-[1-[[3-(trifluoromethyl)phenyl]methyl]piperidin-4-yl]acetamide |
CFAMM00131066 |
CHEMBL373491 |
Bioactive |
(2S)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-2-(4-fluorophenyl)-4-[(1S,3'S)-3'-methylspiro[indene-1,4'-piperidine]-1'-yl]butanamide |
CFAMM00131158 |
CHEMBL42972 |
Bioactive |
AGN-PC-073MIP |
CFAMM00131033 |
CHEMBL23880 |
Bioactive |
N-[4-[(1S)-1-amino-2-[(3S)-3-fluoropyrrolidin-1-yl]-2-oxoethyl]cyclohexyl]-2-(trifluoromethyl)benzamide |
CFAMM00131124 |
CHEMBL271752 |
Bioactive |
N-[2-oxo-2-[[(1S,2R)-2-[[4-(trifluoromethyl)phenyl]methylamino]cyclohexyl]amino]ethyl]-3-(trifluoromethyl)benzamide |
CFAMM00131059 |
CHEMBL1829636 |
Bioactive |
N-[2-[[1-(4-fluoro-4-phenylcyclohexyl)azetidin-3-yl]amino]-2-oxoethyl]-3-(trifluoromethyl)benzamide |
CFAMM00131087 |
CHEMBL2031978 |
Bioactive |
AGN-PC-0068HW |
CFAMM00130936 |
CHEMBL413091 |
Bioactive |
AGN-PC-073GMP |
CFAMM00130952 |
CHEMBL386865 |
Bioactive |
(2R)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-2-(4-fluorophenyl)-4-(4-phenylpiperidin-1-yl)butanamide |
CFAMM00131011 |
CHEMBL549514 |
Bioactive |
N-[(3R)-1-[(6-fluoronaphthalen-2-yl)methyl]pyrrolidin-3-yl]-2-phenylacetamide |
CFAMM00131052 |
CHEMBL345305 |
Bioactive |
(2R)-N-[(2S)-3,3-dimethyl-1-oxo-1-[[(1R)-1-phenylethyl]amino]butan-2-yl]-N'-hydroxy-2-[3-[4-phenyl-3-(trifluoromethyl)phenyl]propyl]butanediamide |
CFAMM00131117 |
CHEMBL1092343 |
Bioactive |
SureCN11888280 |
CFAMM00131080 |
CHEMBL69466 |
Bioactive |
AGN-PC-074G5B |
CFAMM00131093 |
CHEMBL104435 |
Bioactive |
3-[[[3,5-bis(trifluoromethyl)phenyl]methylamino]methyl]-2,6,7-trimethyl-4-phenylisoquinolin-1-one |
CFAMM00131143 |
CHEMBL247203 |
Bioactive |
SureCN5113256 |
CFAMM00131045 |
CHEMBL247407 |
Bioactive |
SureCN5126634 |
CFAMM00130984 |
CHEMBL1090548 |
Bioactive |
SureCN13271687 |
CFAMM00131149 |
CHEMBL474018 |
Bioactive |
N-(3-methoxypropyl)-2-phenyl-N-[[2-[4-(piperazin-1-ylmethyl)phenyl]phenyl]methyl]acetamide |
CFAMM00130977 |
CHEMBL556735 |
Bioactive |
(4R,7S,10S,13S,16S,19S)-10-(4-aminobutyl)-19-[[(2S)-2-amino-3-(4-carbamoylphenyl)propanoyl]amino]-N-[(2S)-1-amino-3-naphthalen-2-yl-1-oxopropan-2-yl]-7,16-dibenzyl-13-[methyl(naphthalene-2-carbonyl)amino]-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide |
CFAMM00131079 |
CHEMBL436951 |
Bioactive |
N-[2-[3,5-bis(trifluoromethyl)phenyl]propan-2-yl]-N-methyl-2-phenylbenzamide |
CFAMM00131018 |
CHEMBL2022528 |
Bioactive |
N-[2-[(2S,4S)-2-cyano-4-fluoropyrrolidin-1-yl]-2-oxoethyl]naphthalene-1-carboxamide |
CFAMM00131044 |
CHEMBL425225 |
Bioactive |
(E)-3-phenyl-N-(3-spiro[1,2-dihydroindene-3,4'-piperidine]-1'-ylpropyl)prop-2-enamide |
CFAMM00130957 |
CHEMBL424895 |
Bioactive |
(2S)-1-[[(6S)-6-[[4-(4-fluorophenyl)benzoyl]-methylamino]-5,6,7,8-tetrahydronaphthalen-2-yl]methyl]-N,N-dimethylpyrrolidine-2-carboxamide |
CFAMM00130970 |
CHEMBL552292 |
Bioactive |
N-[(1R)-1-(4-bromophenyl)ethyl]-4-[[1-[(2,4-dimethylphenyl)methyl]piperidin-4-ylidene]methyl]benzamide |
CFAMM00131071 |
CHEMBL246403 |
Bioactive |
SureCN5115486 |
CFAMM00130933 |
CHEMBL1088810 |
Bioactive |
SureCN11888262 |
CFAMM00131024 |
CHEMBL266972 |
Bioactive |
N-[(2R)-5-(diaminomethylideneamino)-1-oxo-1-[[4-(trifluoromethyl)phenyl]methylamino]pentan-2-yl]naphthalene-2-carboxamide |
CFAMM00131037 |
CHEMBL551134 |
Bioactive |
4-fluoro-N-[(3R)-1-[(6-fluoronaphthalen-2-yl)methyl]pyrrolidin-3-yl]benzamide |
CFAMM00130940 |
CHEMBL1089965 |
Bioactive |
SureCN13271618 |
CFAMM00131002 |
CHEMBL401463 |
Bioactive |
SureCN5116341 |
CFAMM00131091 |
CHEMBL1910390 |
Bioactive |
9-[1-(anthracene-9-carbonyl)piperidin-4-yl]-2-ethyl-2,9-diazaspiro[4.5]decan-1-one |
CFAMM00131121 |
CHEMBL528992 |
Bioactive |
N-[(1R,5R)-8-[(6-fluoronaphthalen-2-yl)methyl]-8-azabicyclo[3.2.1]octan-3-yl]-2-(pyrrolidine-1-carbonyl)benzamide |
CFAMM00130956 |
CHEMBL468252 |
Bioactive |
(2S)-2-[(3S)-4-[(2R)-2-amino-3-(4-fluorophenyl)propanoyl]-3-[2-(dimethylamino)ethyl]-2-oxopiperazin-1-yl]-N-methyl-3-naphthalen-2-ylpropanamide |
CFAMM00130969 |
CHEMBL247210 |
Bioactive |
N-[2-[[(2S)-3-[(2,4-dimethylphenyl)methylamino]-1-oxo-1-pyrrolidin-1-ylpropan-2-yl]amino]-2-oxoethyl]-3-(trifluoromethyl)benzamide |
CFAMM00131043 |
CHEMBL562475 |
Bioactive |
N-[(3R)-1-[(6-fluoronaphthalen-2-yl)methyl]pyrrolidin-3-yl]-2-phenylbenzamide |
CFAMM00131008 |
CHEMBL2029406 |
Bioactive |
N-[2-oxo-2-[(3R)-3-[(4-phenylcyclohexyl)amino]pyrrolidin-1-yl]ethyl]-3-(trifluoromethyl)benzamide |
CFAMM00131056 |
CHEMBL212939 |
Bioactive |
AGN-PC-0764WC |
CFAMM00131161 |
CHEMBL213648 |
Bioactive |
(2S)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-4-(3'-ethylspiro[indene-1,4'-piperidine]-1'-yl)-2-(4-fluorophenyl)butanamide |
CFAMM00130975 |
CHEMBL2057752 |
Bioactive |
4-(4-fluorobenzoyl)-N-[(1R,5R)-8-[(6-fluoronaphthalen-2-yl)methyl]-8-azabicyclo[3.2.1]octan-3-yl]-1,4-diazepane-1-carboxamide |
CFAMM00130988 |
CHEMBL50584 |
Bioactive |
AGN-PC-073ROT |
CFAMM00131049 |
CHEMBL462044 |
Bioactive |
SureCN5844834 |
CFAMM00131140 |
CHEMBL247208 |
Bioactive |
SureCN5119346 |
CFAMM00131016 |
CHEMBL488529 |
Bioactive |
N-[(1R,5R)-8-[(6-fluoronaphthalen-2-yl)methyl]-8-azabicyclo[3.2.1]octan-3-yl]-2-(morpholine-4-carbonyl)benzamide |
CFAMM00131090 |
CHEMBL425801 |
Bioactive |
N-[(2R)-5-(diaminomethylideneamino)-1-oxo-1-[[4-(trifluoromethyl)phenyl]methylamino]pentan-2-yl]-4-fluoronaphthalene-1-carboxamide |
CFAMM00131133 |
CHEMBL1090715 |
Bioactive |
(E,2R)-5-(3-fluorophenyl)-2-(naphthalene-2-carbonylamino)pent-4-enoic acid |
CFAMM00130955 |
CHEMBL2057490 |
Bioactive |
N-[3-(4-benzhydrylpiperidin-1-yl)propyl]-6-fluoro-1-oxo-3,4-dihydroisoquinoline-2-carboxamide |
CFAMM00130968 |
CHEMBL247211 |
Bioactive |
N-[2-[[(2S)-3-[(2,4-dimethylphenyl)methylamino]-1-morpholin-4-yl-1-oxopropan-2-yl]amino]-2-oxoethyl]-3-(trifluoromethyl)benzamide |
CFAMM00130981 |
CHEMBL281731 |
Bioactive |
AGN-PC-02X95J |
CFAMM00131083 |
CHEMBL400159 |
Bioactive |
SureCN5125141 |
CFAMM00131146 |
CHEMBL246213 |
Bioactive |
SureCN5115567 |
CFAMM00131160 |
CHEMBL471633 |
Bioactive |
(3R)-3-amino-N-(1-benzyl-4-phenylpiperidin-4-yl)-4-(2-fluorophenyl)butanamide |
CFAMM00131069 |
CHEMBL246401 |
Bioactive |
SureCN5114482 |
CFAMM00130947 |
CHEMBL209975 |
Bioactive |
(2S)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-2-(4-fluorophenyl)-5-piperidin-1-ylpentanamide |
CFAMM00130987 |
CHEMBL379634 |
Bioactive |
(2S)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-4-[(1R,3'R)-3'-ethylspiro[indene-1,4'-piperidine]-1'-yl]-2-(4-fluorophenyl)butanamide |
CFAMM00131061 |
CHEMBL110349 |
Bioactive |
AGN-PC-00KE0H |
CFAMM00131126 |
CHEMBL1089629 |
Bioactive |
N-[2-oxo-2-[[(3R)-1-[2-[1-[4-(trifluoromethyl)benzoyl]piperidin-4-yl]ethyl]pyrrolidin-3-yl]amino]ethyl]-3-(trifluoromethyl)benzamide |
CFAMM00130938 |
CHEMBL2031991 |
Bioactive |
N-[[(3S)-1-[6,6-bis(4-fluorophenyl)hexanoyl]pyrrolidin-3-yl]methyl]-3,5-bis(trifluoromethyl)benzamide |
CFAMM00131089 |
CHEMBL23879 |
Bioactive |
N-[4-[(1S)-1-amino-2-[(3R)-3-fluoropyrrolidin-1-yl]-2-oxoethyl]cyclohexyl]-2-(trifluoromethyl)benzamide |
CFAMM00131166 |
CHEMBL248423 |
Bioactive |
SureCN5125169 |
CFAMM00130980 |
CHEMBL192354 |
Bioactive |
(2S)-4-benzoyl-N-benzyl-1-[(2S)-5-(diaminomethylideneamino)-2-[(2-naphthalen-2-ylacetyl)amino]pentanoyl]piperazine-2-carboxamide |
CFAMM00131041 |
CHEMBL51588 |
Bioactive |
AGN-PC-073RQE |
CFAMM00131119 |
CHEMBL410829 |
Bioactive |
N-[2-[[(3R)-1-benzylpyrrolidin-3-yl]amino]-2-oxoethyl]-3-(trifluoromethyl)benzamide |
CFAMM00131159 |
CHEMBL1093153 |
Bioactive |
SureCN11888271 |
CFAMM00130993 |
CHEMBL2409074 |
Bioactive |
(E,3R)-6-(3-fluorophenyl)-3-(naphthalene-2-carbonylamino)hex-5-enoic acid |
CFAMM00131006 |
CHEMBL1682658 |
Bioactive |
(1S,2R)-2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-N-[(4-fluorophenyl)methyl]-N-methyl-1-[3-(trifluoromethyl)phenyl]cyclopropane-1-carboxamide |
CFAMM00131108 |
CHEMBL200270 |
Bioactive |
3-[[[2-[[(2S)-2-[[(2R)-2-[[1-(butanoylamino)-4-phenylcyclohexanecarbonyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-naphthalen-2-ylpropanoyl]amino]methyl]benzamide |
CFAMM00131021 |
CHEMBL2348281 |
Bioactive |
N-(1-butyl-5,6-dimethyl-2-oxopyridin-3-yl)naphthalene-2-carboxamide |
CFAMM00131138 |
CHEMBL530560 |
Bioactive |
2-(azepane-1-carbonyl)-N-[(1R,5R)-8-[(6-fluoronaphthalen-2-yl)methyl]-8-azabicyclo[3.2.1]octan-3-yl]benzamide |
CFAMM00130986 |
CHEMBL518772 |
Bioactive |
AGN-PC-0791CJ |
CFAMM00131047 |
CHEMBL535180 |
Bioactive |
(3R)-3-amino-1-(2-benzoyldiazinan-1-yl)-4-(2,4,5-trifluorophenyl)butan-1-one;hydrochloride |
CFAMM00131013 |
CHEMBL439062 |
Bioactive |
N-[2-[[(3R)-1-[(2-naphthalen-2-ylphenyl)methyl]pyrrolidin-3-yl]amino]-2-oxoethyl]-3-(trifluoromethyl)benzamide |
CFAMM00131101 |
CHEMBL90129 |
Bioactive |
AC1LAK9W |
CFAMM00130979 |
CHEMBL337246 |
Bioactive |
Teijin-lead_cmp_5 |
CFAMM00131118 |
CHEMBL492802 |
Bioactive |
4-cyano-N-[[3-[3-(piperazin-1-ylmethyl)phenyl]phenyl]methyl]benzamide |
CFAMM00130966 |
CHEMBL499971 |
Bioactive |
2-N-cyclohexyl-1-N-[(1R,5R)-8-[(6-fluoronaphthalen-2-yl)methyl]-8-azabicyclo[3.2.1]octan-3-yl]-2-N-methylbenzene-1,2-dicarboxamide |
CFAMM00131144 |
CHEMBL247205 |
Bioactive |
SureCN5111992 |
CFAMM00130959 |
CHEMBL209899 |
Bioactive |
(2S)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-2-(4-fluorophenyl)-4-(4-phenylpiperidin-1-yl)butanamide |
CFAMM00131020 |
CHEMBL247207 |
Bioactive |
SureCN5125111 |
CFAMM00131046 |
CHEMBL207462 |
Bioactive |
N-[[4-[[(1S)-2-(cyclopropylmethylamino)-2-oxo-1-phenylethyl]carbamoyl]phenyl]methyl]-2-[4-(trifluoromethyl)phenyl]benzamide |
CFAMM00131094 |
CHEMBL213880 |
Bioactive |
CHEMBL213880 |
CFAMM00131137 |
CHEMBL214770 |
Bioactive |
(2S)-2-[(3S)-3-(2-aminoethyl)-4-[(2R)-2-amino-3-(4-fluorophenyl)propanoyl]-2-oxopiperazin-1-yl]-N-methyl-3-naphthalen-2-ylpropanamide |
CFAMM00131150 |
CHEMBL460349 |
Bioactive |
SureCN5845113 |
CFAMM00131073 |
CHEMBL246407 |
Bioactive |
SureCN5126006 |
CFAMM00131164 |
CHEMBL277635 |
Bioactive |
N-[4-[(1S)-1-amino-2-(3,3-difluoropyrrolidin-1-yl)-2-oxoethyl]cyclohexyl]-2-(trifluoromethyl)benzamide |
CFAMM00130965 |
CHEMBL234643 |
Bioactive |
AGN-PC-0769MQ |
CFAMM00131039 |
CHEMBL261955 |
Bioactive |
N-methyl-N-[(3S)-1-[(3R)-3-(2-phenylethylamino)pyrrolidine-1-carbonyl]pyrrolidin-3-yl]-4-[4-(trifluoromethyl)phenyl]benzamide |
CFAMM00131004 |
CHEMBL522295 |
Bioactive |
AGN-PC-04T7P4 |
CFAMM00131019 |
CHEMBL1829609 |
Bioactive |
N-[2-oxo-2-[[1-(4-phenylcyclohexyl)azetidin-3-yl]amino]ethyl]-3-(trifluoromethyl)benzamide |
CFAMM00130958 |
CHEMBL207369 |
Bioactive |
SureCN6254466 |
CFAMM00130971 |
CHEMBL185866 |
Bioactive |
9-[4-(5-benzamido-2-oxo-1,3,2$l^{5}-dioxaphosphinan-2-yl)butyl]-N-(2,2,2-trifluoroethyl)fluorene-9-carboxamide |
CFAMM00131106 |
CHEMBL517108 |
Bioactive |
SureCN5845214 |
CFAMM00131123 |
CHEMBL213601 |
Bioactive |
(2S)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-2-(4-fluorophenyl)-4-[(1R,3'R)-3'-methylspiro[indene-1,4'-piperidine]-1'-yl]butanamide |
CFAMM00131058 |
CHEMBL92133 |
Bioactive |
AC1LAK9Z |
CFAMM00131136 |
CHEMBL479071 |
Bioactive |
AGN-PC-04TJH7 |
CFAMM00131163 |
CHEMBL215550 |
Bioactive |
N-[(3S)-1-[(3R)-3-(3-cyclohexylpropylamino)pyrrolidine-1-carbonyl]pyrrolidin-3-yl]-N-methyl-4-[4-(trifluoromethyl)phenyl]benzamide |
CFAMM00131086 |
CHEMBL280654 |
Bioactive |
2-[(E)-2-naphthalen-2-ylethenyl]-N-(1-oxo-3-phenylpropan-2-yl)benzamide |
CFAMM00131099 |
CHEMBL2031982 |
Bioactive |
N-[[1-[6,6-bis(4-fluorophenyl)hexyl]pyrrolidin-3-yl]methyl]-3,5-bis(trifluoromethyl)benzamide |
CFAMM00131129 |
CHEMBL452289 |
Bioactive |
4'-[(1r)-1-Amino-2-(2,5-Difluorophenyl)ethyl]biphenyl-3-Carboxamide |
CFAMM00131142 |
CHEMBL1784170 |
Bioactive |
N-cyclopropyl-3-fluoro-5-[4-(2-methoxyethylcarbamoyl)phenyl]-4-methylbenzamide |
CFAMM00130964 |
CHEMBL283475 |
Bioactive |
AGN-PC-037CEI |
CFAMM00131038 |
CHEMBL560198 |
Bioactive |
(E)-N-[(3R)-1-[(6-fluoronaphthalen-2-yl)methyl]pyrrolidin-3-yl]-3-phenylprop-2-enamide |
CFAMM00131051 |
CHEMBL246399 |
Bioactive |
SureCN5116342 |
CFAMM00131156 |
CHEMBL493678 |
Bioactive |
AGN-PC-04WW41 |
CFAMM00130941 |
CHEMBL258996 |
Bioactive |
N-[(1S,5S)-8-[(6-fluoronaphthalen-2-yl)methyl]-8-azabicyclo[3.2.1]octan-3-yl]-2-phenylbenzamide |
CFAMM00131003 |
CHEMBL434609 |
Bioactive |
(E)-5-amino-N-[(2R)-1-[[(2R)-3-(3,4-difluorophenyl)-1-(methylamino)-1-oxopropan-2-yl]-methylamino]-3-naphthalen-2-yl-1-oxopropan-2-yl]-N,5-dimethylhex-2-enamide |
CFAMM00131031 |
CHEMBL1092929 |
Bioactive |
SureCN13271602 |
CFAMM00130996 |
CHEMBL460142 |
Bioactive |
SureCN5846436 |
CFAMM00130950 |
CHEMBL311756 |
Bioactive |
2-[(2S)-3-methyl-2-[[4-(morpholine-4-carbonyl)benzoyl]amino]butanoyl]-N-(5,5,6,6,6-pentafluoro-2-methyl-4-oxohexan-3-yl)-3,4-dihydro-1H-isoquinoline-3-carboxamide |
CFAMM00130963 |
CHEMBL401010 |
Bioactive |
SureCN5126052 |
CFAMM00131009 |
CHEMBL2029408 |
Bioactive |
N-[2-[(3S)-3-[methyl-(4-phenylcyclohexyl)amino]pyrrolidin-1-yl]-2-oxoethyl]-3-(trifluoromethyl)benzamide |
CFAMM00131085 |
CHEMBL377227 |
Bioactive |
N-[[4-[[(1S)-2-oxo-1-phenyl-2-(propylamino)ethyl]carbamoyl]phenyl]methyl]-2-[4-(trifluoromethyl)phenyl]benzamide |
CFAMM00131098 |
CHEMBL214747 |
Bioactive |
AGN-PC-0764VF |
CFAMM00130976 |
CHEMBL93625 |
Bioactive |
AC1LAK9T |
CFAMM00130989 |
CHEMBL290926 |
Bioactive |
1-[(2R,4S)-2-benzyl-1-[3,5-bis(trifluoromethyl)benzoyl]piperidin-4-yl]-3-propan-2-ylurea |
CFAMM00131063 |
CHEMBL515848 |
Bioactive |
Smac mimetic, 8 |
CFAMM00131141 |
CHEMBL247209 |
Bioactive |
N-[2-[[(2S)-3-[(2,4-dimethylphenyl)methylamino]-1-oxo-1-(2,2,2-trifluoroethylamino)propan-2-yl]amino]-2-oxoethyl]-3-(trifluoromethyl)benzamide |
CFAMM00131168 |
CHEMBL80903 |
Bioactive |
2-[(E)-2-naphthalen-1-ylethenyl]-N-(1-oxo-3-phenylpropan-2-yl)benzamide |
CFAMM00131104 |
CHEMBL380666 |
Bioactive |
N-[[4-[[(1S)-2-[butyl(methyl)amino]-2-oxo-1-phenylethyl]carbamoyl]phenyl]methyl]-2-[4-(trifluoromethyl)phenyl]benzamide |
CFAMM00131134 |
CHEMBL460138 |
Bioactive |
SureCN5843458 |
CFAMM00130982 |
CHEMBL330860 |
Bioactive |
(E)-5-amino-N-[(2R)-1-[[(2R)-1-(ethylamino)-1-oxo-3-phenylpropan-2-yl]-methylamino]-3-naphthalen-2-yl-1-oxopropan-2-yl]-N,5-dimethylhex-2-enamide |
CFAMM00130995 |
CHEMBL1779690 |
Bioactive |
4-[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butanoyl]-1-[(4-phenylphenyl)methyl]piperazin-2-one |
CFAMM00131036 |
CHEMBL476557 |
Bioactive |
SureCN2007259 |
CFAMM00130939 |
CHEMBL2069842 |
Bioactive |
(3R)-3-amino-1-[4-[4-(trifluoromethyl)benzoyl]piperazin-1-yl]-4-(2,4,5-trifluorophenyl)butan-1-one |
CFAMM00131103 |
CHEMBL213835 |
Bioactive |
N-methyl-N-[(3S)-1-[(3S)-3-(3-phenylpropylamino)pyrrolidine-1-carbonyl]pyrrolidin-3-yl]-4-[4-(trifluoromethyl)phenyl]benzamide |
CFAMM00131120 |
CHEMBL427522 |
Bioactive |
AGN-PC-075FRJ |
CFAMM00130994 |
CHEMBL1823353 |
Bioactive |
N-[4-[4-[2-(ethylamino)-2-oxo-1-phenylethyl]piperazin-1-yl]-3-fluorophenyl]-2-phenylbenzamide |
CFAMM00131007 |
CHEMBL2029407 |
Bioactive |
N-[2-oxo-2-[(3S)-3-[(4-phenylcyclohexyl)amino]pyrrolidin-1-yl]ethyl]-3-(trifluoromethyl)benzamide |
CFAMM00131035 |
CHEMBL477557 |
Bioactive |
AGN-PC-077L2M |
CFAMM00130961 |
CHEMBL385824 |
Bioactive |
(2S)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-2-(4-fluorophenyl)-4-(3'-methylspiro[indene-1,4'-piperidine]-1'-yl)butanamide |
CFAMM00131139 |
CHEMBL277279 |
Bioactive |
(2S)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-2-(4-fluorophenyl)-4-spiro[indene-1,4'-piperidine]-1'-ylbutanamide |
CFAMM00130954 |
CHEMBL2057491 |
Bioactive |
N-[(1R,5R)-8-[(6-fluoronaphthalen-2-yl)methyl]-8-azabicyclo[3.2.1]octan-3-yl]-2-phenylbenzamide |
CFAMM00131000 |
CHEMBL246415 |
Bioactive |
N-[2-[[(2S)-1-(tert-butylamino)-3-[(2,4-dimethylphenyl)methylamino]-1-oxopropan-2-yl]amino]-2-oxoethyl]-3-(1,1,2,2,2-pentafluoroethyl)benzamide |
CFAMM00131028 |
CHEMBL400196 |
Bioactive |
SureCN5128373 |
CFAMM00131075 |
CHEMBL394189 |
Bioactive |
N-[4-(4-benzhydryl-1,4-diazepan-1-yl)butyl]naphthalene-2-carboxamide |
CFAMM00131152 |
CHEMBL184551 |
Bioactive |
AGN-PC-075FPK |
CFAMM00131054 |
CHEMBL1162933 |
Bioactive |
CHEMBL1162933 |
CFAMM00131068 |
CHEMBL382273 |
Bioactive |
4-[[[2-[[(2S)-2-[[(2R)-2-[[1-(butanoylamino)-4-phenylcyclohexanecarbonyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-naphthalen-2-ylpropanoyl]amino]methyl]benzamide |
CFAMM00131145 |
CHEMBL247206 |
Bioactive |
SureCN5120132 |
CFAMM00130960 |
CHEMBL202715 |
Bioactive |
AGN-PC-00CSNO |
CFAMM00131040 |
57323835 |
Patent Compound |
AGN-PC-0BR9XU |
CFAMM00131053 |
15383377 |
Patent Compound |
AGN-PC-00P2JZ |
CFAMM00130972 |
12942329 |
Patent Compound |
AGN-PC-00K6JT |
CFAMM00131107 |
53731786 |
Patent Compound |
AGN-PC-09Y293 |
CFAMM00131025 |
54360861 |
Patent Compound |
SureCN6318694 |
CFAMM00131113 |
54371801 |
Patent Compound |
|
CFAMM00131112 |
54251940 |
Patent Compound |
SureCN7598989 |
CFAMM00131050 |
53935945 |
Patent Compound |
|
CFAMM00131078 |
57077124 |
Patent Compound |
|
CFAMM00131084 |
9851153 |
Patent Compound |
SureCN8397653 |
CFAMM00130962 |
18794521 |
Patent Compound |
AGN-PC-022LQV |
CFAMM00131097 |
54006412 |
Patent Compound |
SureCN8174212 |
CFAMM00131111 |
54378273 |
Patent Compound |
AGN-PC-0A66NV |
CFAMM00131062 |
18794666 |
Patent Compound |
AGN-PC-022LUF |
CFAMM00131127 |
53832921 |
Patent Compound |
|
CFAMM00131076 |
18794713 |
Patent Compound |
AGN-PC-022LVJ |
CFAMM00131167 |
53759916 |
Patent Compound |
AGN-PC-030FIS |
CFAMM00131029 |
54180911 |
Patent Compound |
SureCN8426019 |
CFAMM00131055 |
53732112 |
Patent Compound |
SureCN7650999 |
CFAMM00131109 |
54535786 |
Patent Compound |
SureCN7647106 |
CFAMM00131022 |
57082124 |
Patent Compound |
|
CFAMM00131048 |
53657672 |
Patent Compound |
SureCN6326308 |
CFAMM00131082 |
10673683 |
Patent Compound |
SureCN6320599 |
CFAMM00131034 |
53838051 |
Patent Compound |
SureCN8170106 |